859230-84-5
Chemical Structure
BMS-505130 fumarate
- CAS No.: 859230-84-5
- Formula:C19H21N3O4
- Molecular Weight:355.39
IUPAC Name: 3-((1S,2S)-2-((dimethylamino)methyl)cyclopropyl)-1H-indole-5-carbonitrile maleate
InChIKey: QYXJWBDKQAIHJM-ZMPXXIOZSA-N
SMILES: O=C(O)/C=C\C(O)=O.CN(C)C[C@@H]1[C@@H](C2=CNC3=CC=C(C#N)C=C23)C1
Biological Activity: BMS-505130 fumarate is a potent, selective and orally active serotonin transport inhibitor with a Ki for binding to the serotonin transporter of 0.18 nM (Ki for norepinephrine and dopamine transporters of 4.6 and 2.1 μM, respectively). BMS-505130 fumarate can be used for the research of neurological disease, such as depression[1].
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BMS-505130 fumarate | BMS-505130 fumarate is a potent, selective and orally active serotonin transport inhibitor with a Ki for binding to the serotonin transporter of 0.18 nM (Ki for norepinephrine and dopamine transporters of 4.6 and 2.1 μM, respectively). BMS-505130 fumarate can be used for the research of neurological disease, such as depression. | |||||||||||||||||||||
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Keywords
