90808-12-1
90808-12-1
Chemical Structure
Divaplon
Synonym(s): RU 32698
- CAS No.: 90808-12-1
- Formula:C17H17N3O2
- Molecular Weight:295.34
IUPAC Name: (6-ethyl-7-methoxy-5-methylimidazo[1,2-a]pyrimidin-2-yl)(phenyl)methanone
InChIKey: NRJVHCSYLGLURI-UHFFFAOYSA-N
SMILES: O=C(C1=CN2C(C)=C(CC)C(OC)=NC2=N1)C3=CC=CC=C3
Biological Activity: Divaplon is a GABA receptor agonist with the EC50 values of 31 and 2 nM for α3β2γ2 and α5β2γ2, respectively. Divaplon shows anxiolytic activity[1][2].
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Divaplon | Divaplon is a GABA receptor agonist with the EC50 values of 31 and 2 nM for α3β2γ2 and α5β2γ2, respectively. Divaplon shows anxiolytic activity. | |||||||||||||||||||||
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References
- [1]. Knoflach F, et al. Full and partial agonism displayed by benzodiazepine receptor ligands at recombinant gamma-aminobutyric acidA receptor subtypes. J Pharmacol Exp Ther. 1993;266(1):385-391. [Content Brief]
- [2]. Sanger DJ, et al. Benzodiazepine (omega) receptor partial agonists and the acquisition of conditioned fear in mice. Psychopharmacology (Berl). 1995;121(1):104-108. [Content Brief]
Keywords
