GNE-1567
GNE-1567 is a potent ERα PROTAC degrader and a selective XIAP antagonist with a Kd value of 0.03 μM. GNE-1567 is indicated for breast cancer research.
(Pink: ERα ligand (HY-18719); Blue: XIAP ligand (HY-175449); Black: linker).
Para uso exclusivo en investigación. No vendemos a pacientes.
- Fòrmula: C60H65BrN6O9
- Peso molecular:1094.10
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Ver todos los productos específicos de isoformas PROTACs
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Actividad biológica
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XIAP 0.03 μM (Kd) |
Chemical Information
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Peso molecular 1094.10
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Fòrmula C60H65BrN6O9
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SMILES
CC/C(C1=CC=CC=C1)=C(C2=CC=C(O)C=C2)/C3=CC=C(C=C3)OCCN(C(CCOCCOCCC(N4C5=C(N(C([C@H]([C@@H]4C)NC([C@@H](NC)C)=O)=O)CC6=C(C=CC7=C6C=CC(Br)=C7)OC)C=CC(C#N)=C5)=O)=O)C
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)