1. Signaling Pathways
  2. Apoptosis
  3. IAP
  4. IAP Inhibitors

IAP Inhibitors

cIAP

cIAP-1

cIAP-2

XIAP

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

IAP Inhibitors, Antagonists, Modulators, Inducers, Degraders & Ligands
Product Name cIAP cIAP-1 cIAP-2 XIAP Purity
SM-164  
cIAP-1, Ki: 0.31 nM
cIAP-2, Ki: 1.1 nM
  99.53%
AZD5582  
cIAP1, IC50: 15 nM
cIAP2, IC50: 21 nM
XIAP, IC50: 15 nM
99.61%
Anticancer agent 294  
cIAP-1, IC50: 15 nM
   
Xevinapant  
cIAP1, Ki: 1.9 nM
cIAP2, Ki: 5.1 nM
XIAP, Ki: 66.4 nM
99.91%
Embelin      
XIAP, IC50: 4.1 μM
99.01%
Jolkinolide B  
cIAP-1
cIAP-2
XIAP
99.65%
SM-164 hydrochloride  
cIAP-1, Ki: 0.31 nM
cIAP-2, Ki: 1.1 nM
 
Xevinapant hydrochloride  
cIAP1, Ki: 1.9 nM
cIAP2, Ki: 5.1 nM
XIAP, Ki: 66.4 nM
98.11%
AZD5582 dihydrochloride  
cIAP1, IC50: 15 nM
cIAP2, IC50: 21 nM
XIAP, IC50: 15 nM
99.92%
TD1092  
cIAP1
cIAP2
XIAP
99.49%
PBX-7016      
XIAP
SBP-0636457      
XIAP, Ki: 0.27 μM
98.42%
Nurr1 agonist 14      
XIAP
99.42%
Bestatin methyl ester
cIAP
     
CDK9-IN-45      
XIAP
KHS108-MV1  
cIAP1
cIAP2
XIAP
HM90822  
cIAP-1
cIAP2
XIAP
ZLMT-72      
XIAP
PROTAC TEAD1/IAP degrader-1  
cIAP1, DC50: 270 nM
   
SM-122  
cIAP-1
cIAP-2
 
Topo I/DDX5-IN-1      
XIAP
GNE-5472    
cIAP-2
 
XIAP ligand-Linker Conjugate 1      
XIAP
Ciapavir
cIAP
     
TP-110  
cIAP-1
 
XIAP
LSD1-IN-26  
cIAP-1
   
Topoisomerase I inhibitor 17      
XIAP
XIAP ligand-Linker Conjugate 2      
XIAP
XIAP/cIAP1 antagonist-1  
cIAP1, IC50: 0.32 nM
 
XIAP, IC50: 5.1 nM
PROTAC EZH2 Degrader-21
cIAP
     
PROTAC EZH2 Degrader-41
cIAP
     
K882      
XIAP
CSLP43      
XIAP
(2''S)-2'',3''-Dihydrodelicaflavone      
XIAP
IAP ligand 9  
cIAP-1
 
XIAP
XIAP ligand 5      
XIAP
IAP ligand 8  
cIAP-1
 
XIAP
GNE-1567      
XIAP, Kd: 0.03 μM
T-3256336  
cIAP1, IC50: 1.3 nM
 
XIAP, IC50: 200 nM
Jolkinolide B (Standard)  
cIAP-1
cIAP-2
XIAP
XB2M54      
XIAP
PROTAC TEAD1/IAP degrader-2
cIAP