CPI-1328
CPI-1328 is an EZH2 inhibitor with a Ki value of 63 fM.
Para uso exclusivo en investigación. No vendemos a pacientes.
- No. CAS: 2390367-27-6
- Fòrmula: C28H36ClN3O4S
- Peso molecular:546.12
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Ver todos los productos específicos de isoformas Histone Methyltransferase
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Actividad biológica
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EZH2 |
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Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HeLa | EC50 |
0.849 nM
Compound: 83
|
Antiproliferative activity against human HeLa cells
Antiproliferative activity against human HeLa cells
|
[PMID: 35531606] |
| KARPAS-422 | GI50 |
5.7 nM
Compound: 83
|
Antiproliferative activity against human KARPAS-422 cells assessed as inhibition of cell growth
Antiproliferative activity against human KARPAS-422 cells assessed as inhibition of cell growth
|
[PMID: 35531606] |
Chemical Information
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No. CAS 2390367-27-6
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Peso molecular 546.12
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Fòrmula C28H36ClN3O4S
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SMILES
ClC1=C2C(O[C@](O2)([C@]3([H])CC[C@H](CC3)N(C)C)C)=C(C4=C1CCN(C4=O)CC5=C(C=C(NC5=O)C)SC)C
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)