JYL 1511
JYL 1511 is a partial agonist of vanilloid receptor VR1.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 623166-14-3
- 分子式: C21H29N3O3S2
- 分子量:435.60
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Help & FAQs
生物活性
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
32.4 nM
Compound: 3
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Agonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assay
Agonist activity at rat TRPV1 expressed in CHO cells by 45Ca2+ uptake assay
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[PMID: 18406014] |
JYL 1511 inhibits [3H]Resiniferatoxin binding to rat VR1 with a Ki of 50.4 nM[1].
JYL 1511 inhibits Capsaicin induction of 45Ca2+ uptake in CHO cells overexpressing rat VR1 (IC50: 3.4 nM)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 623166-14-3
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分子量 435.60
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分子式 C21H29N3O3S2
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SMILES
CS(=O)(NC1=CC=C(C=C1OC)CNC(NCC2=CC=C(C=C2)C(C)(C)C)=S)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
JYL 1511 関連分類
HY-118299 関連分類
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