1. GPCR/G Protein
    Neuronal Signaling
  2. mGluR
  3. MPEP

MPEP 

Cat. No.: HY-14609A
Handling Instructions

MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.

For research use only. We do not sell to patients.

MPEP Chemical Structure

MPEP Chemical Structure

CAS No. : 96206-92-7

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50 mg USD 276 Ask For Quote & Lead Time

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Description

MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors. IC50 value: 36 nM Target: mGluR5 Centrally active following systemic administration in vivo. Reverses mechanical hyperalgesia in the inflamed rat hind paw.

Molecular Weight

193.24

Formula

C₁₄H₁₁N

CAS No.

96206-92-7

SMILES

CC1=NC(C#CC2=CC=CC=C2)=CC=C1

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

MPEPmGluRMetabotropic glutamate receptorsInhibitorinhibitorinhibit

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MPEP
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