Discovery of a potent, orally active, nonsteroidal androgen receptor agonist: 4-ethyl-1,2,3,4-tetrahydro-6- (trifluoromethyl)-8-pyridono[5,6-g]- quinoline (LG121071)

  • J Med Chem. 1999 Jan 28;42(2):210-2. doi: 10.1021/jm9806648.
L G Hamann  1 ,  N S Mani ,  R L Davis ,  X N Wang ,  K B Marschke ,  T K Jones
Affiliations
  • 1. Departments of Medicinal Chemistry, Endocrine Research, and New Leads Discovery, Ligand Pharmaceuticals, Inc., 10275 Science Center Drive, San Diego, California 92121, USA. [email protected]
PMID: 9925725 DOI: 10.1021/jm9806648