1 Result for "

2216703-12-5

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "2216703-12-5" in MCE Product Catalog:

Cat. No.: HY-130245A
CAS No.: 2216703-12-5
Target:  

HyT PCSK9

(R,R)-PCSK9 degrader 1 is an isomer of PCSK9 degrader 1 (HY-130245). (R,R)-PCSK9 degrader 1 is a HyT-like PCSK9 degrader (IC50 of 655.4 nM) , and its PCSK9-binding site does not interfere with the binding of PCSK9 to LDL receptor. (R,R)-PCSK9 degrader 1 can be used in the research of atherosclerosis, hypercholesterolemia, coronary heart disease, metabolic syndrome, acute coronary syndrome, and related cardiovascular and cardiometabolic diseases .
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