1 Result for "

CP 526555-15N,13C,d2

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "CP 526555-15N,13C,d2" in MCE Product Catalog:

Cat. No.: HY-10019S1
Synonyms: CP 526555-15N,13C,d2
Varenicline- 15N, 13C,d2 is 15N and deuterated labeled Varenicline (HY-10019). Varenicline (CP 526555) is an orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50=250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of α6β2 nAChR and a full agonist of α7β2 nAChR. Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation .
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