2 Results for "

EGFR-IN-183

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "EGFR-IN-183" in MCE Product Catalog:

Cat. No.: HY-179039
Target:  

EGFR

Research Areas:  

Cancer

EGFR-IN-183 (Compound 5q) is an EGFR inhibitor. EGFR-IN-183 strongly binds to EGFR (T790M/L858R) mutants. EGFR-IN-183 exhibits anti-proliferative activity against MDA-MB-231, with an IC50 value of 16.4 μM. EGFR-IN-183 can be used for research on triple-negative breast cancer .
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Cat. No.: HY-178157
CAS No.: 301820-47-3
Target:  

CDK EGFR VEGFR

Research Areas:  

Cancer

Multi-target kinase-IN-7 (Compound 1e) is an orally active multi-target kinase inhibitor (IC50 values: CDK2=0.314 μM, EGFR=0.183 μM, HER-2=0.197 μM, VEGFR-2=0.235 μM). Multi-target kinase-IN-7 is promising for research of solid tumors (e.g., lung, breast, prostate cancer) .
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