2 Results for "

Ezlopitant

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Ezlopitant" in MCE Product Catalog:

Cat. No.: HY-106982
CAS No.: 147116-64-1
Synonyms: CJ-11,974
Ezlopitant (CJ-11,974) is a selective, non-peptidic neurokinin-1 (NK-1)-receptor antagonist. Ezlopitant inhibits both acute and delayed emetic reactions induced by Cisplatin (HY-17394) in ferrets via acting on NK1 receptors in the central nervous system. Ezlopitant has the potential for pain, chemotherapy-induced emesis and irritable bowel syndrome research .
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Cat. No.: HY-171185
CAS No.: 368454-88-0
Target:  

Drug Metabolite

Research Areas:  

Others

CP-611,781 is a diol metabolite of ezlopitant alkene (CJ-12,458). In human liver microsomes, the apparent KM value of 5.4 μM for the formation of CP-611,781 .
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