1 Result for "

KDM5A-IN-1 (Standard)

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "KDM5A-IN-1 (Standard)" in MCE Product Catalog:

Cat. No.: HY-100014R
CAS No.: 1905481-36-8
Research Areas:  

Cancer

KDM5A-IN-1 (Standard) is the analytical standard of KDM5A-IN-1 (HY-100014). This product is intended for research and analytical applications. KDM5A-IN-1 is a potent, orally bioavailable pan-histone lysine demethylases 5 (KDM5) inhibitor with IC50s of 45 nM, 56 nM and 55 nM for KDM5A, KDM5B and KDM5C, respectively, and with an EC50 value of 960 nM for PC9 H3K4Me3. KDM5A-IN-1 is significantly less potent against other KDM5B enzymes (1A, 2B, 3B, 4C, 6A, 7B) .
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