1 Result for "

Leucettinib92

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "Leucettinib92" in MCE Product Catalog:

Cat. No.: HY-155723
CAS No.: 2732859-57-1
Purity:  98.54%
Target:  

CDK DYRK

Research Areas:  

Others

Leucettinib-92 (compound 92) is an inhibitor of DYRK/CLK kinase, The IC50s are 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 μM (DYRK2), respectively. 1.0 μM (DYRK3), 0.52 μM (DYRK4), 2.78 μM (GSK3) .
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