30 Results for "

N-desethyl

" in MedChemExpress (MCE) Product Catalog:
Products (30)

30 Results for "N-desethyl" in MCE Product Catalog:

6
6 Publications Verification
Cat. No.: HY-10873
CAS No.: 356068-97-8
Purity:  99.90%
Synonyms: SU-12662
Target:  

Drug Metabolite

Research Areas:  

Cancer

N-Desethyl Sunitinib (SU-12662) is a metabolite of Sunitinib (HY-10255A). N-Desethyl Sunitinib serves as a good transport substrate for human ABCB1, ABCG2 and murine ABCG2 .
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6
6 Publications Verification
Cat. No.: HY-138813
Purity:  99.14%
Synonyms: SU-12662 hydrochloride
Target:  

Drug Metabolite

Research Areas:  

Cancer

N-Desethyl Sunitinib (SU-12662) (hydrochloride) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Ki values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively .
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1
1 Cited Publications
Cat. No.: HY-128554
CAS No.: 79352-78-6
Purity:  99.98%
Target:  

Parasite

Research Areas:  

Infection

N-Desethyl amodiaquine is the biologically active metabolite of Amodiaquine (HY-B1322A). N-Desethyl amodiaquine is an antiparasitic agent, has inhibitory for strains V1/S and 3D7 with IC50 values of 97 nM and 25 nM, respectively. N-Desethyl amodiaquine can be used for the research of malaria .
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1
1 Cited Publications
Cat. No.: HY-128554A
CAS No.: 79049-30-2
Purity:  99.45%
Target:  

Parasite

Research Areas:  

Infection

N-Desethyl amodiaquine dihydrochloride is the biologically active metabolite of Amodiaquine (HY-B1322A). N-Desethyl amodiaquine dihydrochloride is an antiparasitic agent, has inhibitory for strains V1/S and 3D7 with IC50 values of 97 nM and 25 nM, respectively. N-Desethyl amodiaquine dihydrochloride can be used for the research of malaria .
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Cat. No.: HY-134124
CAS No.: 92614-59-0
Purity:  95.8%
Research Areas:  

Metabolic Disease

Glutathione ethyl ester is a cell-permeable GSH donor and provides an efficient supply of GSH to the oocyte. Glutathione ethyl ester shows positive effect on the in vitro production of embryos by enhancement of the antioxidative defense .
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Cat. No.: HY-128554S
CAS No.: 1173023-19-2
Purity:  ≥98.0%
N-Desethyl amodiaquine-d5 is the deuterium labeled N-Desethyl amodiaquine. N-Desethyl amodiaquine is the major biologically active metabolite of Amodiaquine. N-Desethyl amodiaquine is an antiparasitic agent. IC50 values for strains V1/S and 3D7 are 97 nM and 25 nM, respectively .
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Cat. No.: HY-128554S1
CAS No.: 1216894-33-5
Purity:  98.76%
N-Desethyl amodiaquine-d5 dihydrochloride is the deuterium labeled N-Desethyl amodiaquine dihydrochloride. N-Desethyl amodiaquine dihydrochloride is the major biologically active metabolite of Amodiaquine. N-Desethyl amodiaquine dihydrochloride is an antiparasitic agent. IC50 values for strains V1/S and 3D7 are 97 nM and 25 nM, respectively .
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Cat. No.: HY-10873S
CAS No.: 1217247-62-5
N-Desethyl Sunitinib-d5 is the deuterium labeled N-Desethyl Sunitinib. N-Desethyl Sunitinib (SU-12662) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Ki values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively .
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Cat. No.: HY-B0191C
CAS No.: 155205-89-3
Target:  

Drug Metabolite

Research Areas:  

Others

N-Desethyl Bimatoprost is a N-desethyl metabolite of Bimatoprost (HY-B0191) .
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Cat. No.: HY-128554AR
CAS No.: 79049-30-2
Research Areas:  

Infection

N-Desethyl amodiaquine dihydrochloride (Standard) is the analytical standard of N-Desethyl amodiaquine dihydrochloride. This product is intended for research and analytical applications. N-Desethyl amodiaquine dihydrochloride is the biologically active metabolite of Amodiaquine (HY-B1322A). N-Desethyl amodiaquine dihydrochloride is an antiparasitic agent, has inhibitory for strains V1/S and 3D7 with IC50 values of 97 nM and 25 nM, respectively. N-Desethyl amodiaquine dihydrochloride can be used for the research of malaria .
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Cat. No.: HY-129903R
CAS No.: 448184-46-1
Research Areas:  

Others

N-Desethyl vardenafil (Standard) is the analytical standard of N-Desethyl vardenafil. This product is intended for research and analytical applications. N-Desethyl vardenafil is the major metabolite of Vardenafil (HY-B0442) and can be detected in human urine .
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Cat. No.: HY-129903S
CAS No.: 1184985-26-9
N-Desethyl Vardenafil-d8 is deuterium labeled N-Desethyl vardenafil.
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Cat. No.: HY-W707566
N-Desethyl sunitinib-d4 maleate is the deuterium labeled N-Desethyl sunitinib maleate.
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Cat. No.: HY-135407S
CAS No.: 1173018-49-9
N-Desethyl Oxybutynin-d5 (hydrochloride) is deuterium labeled N-Desethyl Oxybutynin hydrochloride. N-Desethyl Oxybutynin is the the active metabolite Oxybutynin. Oxybutynin is an anticholinergic agent that inhibits voltage-dependent K+ channels .
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Cat. No.: HY-129903
CAS No.: 448184-46-1
Target:  

Drug Metabolite

Research Areas:  

Others

N-Desethyl vardenafil is the major metabolite of Vardenafil (HY-B0442) and can be detected in human urine .
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Cat. No.: HY-139517S1
CAS No.: 2747914-26-5
N-Desethyl etifoxine-- 13C,d3 is the 13C- and deuterium labeled N-Desethyl etifoxine .
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Cat. No.: HY-10873R
CAS No.: 356068-97-8
Synonyms: SU-12662 (Standard)
Research Areas:  

Cancer

N-Desethyl Sunitinib (Standard) is the analytical standard of N-Desethyl Sunitinib. This product is intended for research and analytical applications. N-Desethyl Sunitinib (SU-12662) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Ki values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively[1].
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Cat. No.: HY-10873S2
CAS No.: 1261432-14-7
Synonyms: SU-12662-d5 hydrochloride
N-Desethyl Sunitinib-d5 (hydrochloride) is a deuterated labeled N-Desethyl Sunitinib . N-Desethyl Sunitinib (SU-12662) is a metabolite of sunitinib. Sunitinib is a potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor with Ki values of 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT, respectively .
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Cat. No.: HY-10873S1
CAS No.: 2012601-57-7
Synonyms: SU-12662-d4 TFA
N-Desethyl Sunitinib-d4 (SU-12662-d4) TFA is deuterium-labeled N-Desethyl Sunitinib (HY-10873) .
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Cat. No.: HY-137966A
CAS No.: 2775292-24-3
Synonyms: AL-8520 oxalate
Target:  

Carbonic Anhydrase

Research Areas:  

Cancer

N-Desethyl Brinzolamide oxalate is a dual inhibitor of Carbonic anhydrase II and Carbonic anhydrase IV with IC50s of 1.28 and 128 nM, respectively .
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