11 Results for "

PAF-AN-1

" in MedChemExpress (MCE) Product Catalog:
Products (11)

11 Results for "PAF-AN-1" in MCE Product Catalog:

Cat. No.: HY-U00040
CAS No.: 115621-84-6
PAF-AN-1 is a platelet activating factor receptor (PAF) antagonist.
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2 Cited Publications
Cat. No.: HY-13511A
CAS No.: 182349-12-8
Purity:  98.77%
Synonyms: UR-12592 Fumarate
Research Areas:  

Inflammation/Immunology

Rupatadine (UR-12592) Fumarate is a potent, orally active and long-lasting dual PAF/H1 antagonist, with Kis of 0.55 μM and 0.1 μM, respectively. Rupatadine Fumarate can be used for the research of allergic rhinitis and urticaria [1] .
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2 Cited Publications
Cat. No.: HY-13511
CAS No.: 158876-82-5
Purity:  99.70%
Synonyms: UR-12592
Research Areas:  

Inflammation/Immunology

Rupatadine (UR-12592) is a potent, orally active and long-lasting dual PAF/H1 antagonist, with Kis of 0.55 μM and 0.1 μM, respectively. Rupatadine can be used for the research of allergic rhinitis and urticaria [1] .
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Cat. No.: HY-13511AR
CAS No.: 182349-12-8
Synonyms: UR-12592 Fumarate (StANdard)
Rupatadine (Fumarate) (Standard) is the analytical standard of Rupatadine (Fumarate). This product is intended for research and analytical applications. Rupatadine (UR-12592) Fumarate is a potent, orally active and long-lasting dual PAF/H1 antagonist, with Kis of 0.55 μM and 0.1 μM, respectively. Rupatadine Fumarate can be used for the research of allergic rhinitis and urticaria [1] .
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Cat. No.: HY-101263
CAS No.: 96801-55-7
Purity:  ≥99.0%
Research Areas:  

Others

2-Thio-PAF, a synthetic analog of PAF, is used in a colorimetric assay for PAF acetylhydrolases .
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Cat. No.: HY-W713925
CAS No.: 89019-63-6
Diheptanoyl Thio-PC is a substrate for all phospholipase A2s (PLA2s) with the exception of cPLA2 and PAF-acetyl hydrolase (PAF-AH).1 Interaction of this compound with a PLA2 results in cleavage of the sn-2 fatty acid generating a free thiol on the lysophospholipid. This free thiol can be detected using chromogenic substrates such as DTNB (Ellman’s reagent) and DTP.
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Cat. No.: HY-106924
CAS No.: 127842-07-3
DF 1111301 is a new antiallergic compound endowed of antihistamine-H1 and anti-PAF activities .
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Cat. No.: HY-13511AS
CAS No.: 1795153-63-7
Synonyms: UR-12592 D4 fumarate
Rupatadine-d4 fumarate is a deuterium labeled Rupatadine fumarate. Rupatadine Fumarate (UR-12592 Fumarate) is a potent dual PAF/H1 antagonist with Ki values of 0.55/0.1 μM (rabbit platelet membranes/guinea pig cerebellum membranes) [1] .
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Cat. No.: HY-13511R
CAS No.: 158876-82-5
Synonyms: UR-12592 (StANdard)
Rupatadine (Standard) is the analytical standard of Rupatadine. This product is intended for research and analytical applications. Rupatadine (UR-12592) is a potent, orally active and long-lasting dual PAF/H1 antagonist, with Kis of 0.55 μM and 0.1 μM, respectively. Rupatadine can be used for the research of allergic rhinitis and urticaria [1] .
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Cat. No.: HY-13511S
Synonyms: UR-12592-d6
Rupatadine-d6 (D-tartrate) is deuterated labeled Rupatadine (HY-13511). Rupatadine (UR-12592) is a potent, orally active and long-lasting dual PAF/H1 antagonist, with Kis of 0.55 μM and 0.1 μM, respectively. Rupatadine can be used for the research of allergic rhinitis and urticaria [1] .
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Cat. No.: HY-182583
CAS No.: 81635-83-8
PAF antagonist-1 is a platelet activating factor (PAF) receptor antagonist with a target Ki of 69 nM. PAF antagonist-1 inhibits PAF binding and displays enhanced affinity at A1, A2 a, and A3 adenosine receptor subtypes compared to related dihydropyridine analogs with smaller ester groups. PAF antagonist-1 can be used for cardiovascular disorders, especially hypertension and coronary heart disease [1].
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