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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
3 Results for "
PROTAC WDR5 degrader 1
" in MedChemExpress (MCE) Product Catalog:
Products (3)
3 Results for "PROTAC WDR5 degrader 1" in MCE Product Catalog:
Cat. No.: HY-168487
CAS No.: 2737222-94-3
PROTAC WDR5 degrader 1 is a heterobifunctional WDR5 PROTAC degrader with a DC50 value of 53 nM and a Kd value of 18 nM, exhibiting selective WDR5 degradation activity and cell permeability. PROTAC WDR5 degrader 1 induces proliferation defects in leukemia cells, with enhanced efficacy in cells overexpressing VHL. PROTAC WDR5 degrader 1 is applicable to research related to acute myeloid leukemia .
Cat. No.: HY-162014
CAS No.: 3032434-45-7
WDR5 degrader-1 is a selective Cereblon-recruiting WDR5 PROTAC degrader. WDR5 degrader-1 induces ubiquitination and degradation of WDR5. WDR5 degrader-1 can be used in the research of pancreatic cancer and leukemia .
Cat. No.: HY-168488
CAS No.: 2737222-78-3
Research Areas:
WDR5 ligand 2 is the ligand for WDR5 and can be used for synthesis of PROTAC WDR5 degrader 1 (HY-168487) .
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