2 Results for "

Rapaglutin A

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Rapaglutin A" in MCE Product Catalog:

Cat. No.: HY-176050
Synonyms: RgA; JW11-D2
Target:  

GLUT

Research Areas:  

Cancer

Rapaglutin A is a glucose transporter (GLUT) inhibitor. Rapaglutin A is a pan-GLUT inhibitor of Class I isoforms GLUT1, GLUT3, and GLUT4 with an IC50 of 12 nM. Rapaglutin A has an inhibitory effect on A549 proliferation .
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Cat. No.: HY-176051
Synonyms: RgE
Target:  

GLUT

Research Areas:  

Cancer

Rapaglutin E (RgE) is a glucose transporter (GLUT) inhibitor. Rapaglutin E exhibits dose-dependent inhibition of [ 3H]-2DG uptake in A549, Jurkat T, PANC10.05, and RBC, with IC50 values 8.9 nM, 3.1 nM, 35.5 nM, 74.2 nM. Rapaglutin E inhibits cell proliferation in A549, PANC10.05, HeLa, Jurkat T, and HEK293T cells .
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