2 Results for "

Tetra-2-pyridinylpyrazine

" in MedChemExpress (MCE) Product Catalog:
Products (2)

2 Results for "Tetra-2-pyridinylpyrazine" in MCE Product Catalog:

Cat. No.: HY-W142632
CAS No.: 25005-97-4
Synonyms: 2,3,5,6-Tetrakis(2-pyridyl)pyrazine
Target:  

MOFs

Research Areas:  

Others

Tetra-2-pyridinylpyrazine (2,3,5,6-Tetrakis(2-pyridyl)pyrazine) is a metal-organic framework (MOF).
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Cat. No.: HY-P12136
CAS No.: 1966181-14-5
Synonyms: FE 205030
Target:  

CGRP Receptor

Research Areas:  

Neurological Disease

Fonagepant (FE 205030) is a calcitonin gene-related peptide (CGRP) receptor antagonist with an IC50 of 0.2 nM. Fonagepant selectively blocks CGRP receptor activity, inhibits CGRP-induced vasodilation, attenuates capsaicin-induced increase in skin blood flow, and blocks CGRP-induced vasodilation in isolated human mesenteric resistance arteries. Fonagepant can be used in studies related to acute migraine attacks .
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