5 Results for "

bibn

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "bibn" in MCE Product Catalog:

47
47 Cited Publications
Cat. No.: HY-10095
CAS No.: 204697-65-4
Purity:  99.83%
Synonyms: bibn-4096; bibn 4096BS
Target:  

CGRP Receptor

Research Areas:  

Neurological Disease

Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP .
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47
47 Cited Publications
Cat. No.: HY-10095A
CAS No.: 586368-06-1
Purity:  99.11%
Synonyms: bibn-4096 hydrochloride; bibn4096BS hydrochloride
Target:  

CGRP Receptor

Research Areas:  

Neurological Disease

Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP .
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Cat. No.: HY-119953
CAS No.: 145301-48-0
Target:  

mAChR

Research Areas:  

Neurological Disease

BIBN-99 is a selective, BBB-penetrable and competitive muscarinic M2 receptor antagonist. BIBN-99 improves cognitive performancein rats with traumatic brain injury .
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Cat. No.: HY-117966
CAS No.: 145301-79-7
Target:  

mAChR

Research Areas:  

Cardiovascular Disease

Bibn 140 is a pyridine derivative substituted with a benzene ring, which has high affinity (Ki: 12 nM) and selectivity for M2 mAChR receptors over M1 receptors .
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Cat. No.: HY-10095R
CAS No.: 204697-65-4
Synonyms: bibn-4096 (Standard); bibn 4096BS (Standard)
Research Areas:  

Neurological Disease

Olcegepant (Standard) is the analytical standard of Olcegepant (HY-10095). This product is intended for research and analytical applications. Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP .
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