9 Results for "

neuromuscular blockade

" in MedChemExpress (MCE) Product Catalog:
Products (9)

9 Results for "neuromuscular blockade" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-B0423
CAS No.: 114-80-7
Synonyms: Eustigmin bromide; Neoserine bromide
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

Neostigmine (Eustigmin) Bromide is an orally active and reversible cholinesterase inhibitor that acts on myasthenia gravis to prolong and intensify the muscarinic and nicotinic effects of acetylcholine. Neostigmine Bromide can be used in anesthesia to reverse the neuromuscular blockade produced by competitive neuromuscular blockers .
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1
1 Cited Publications
Cat. No.: HY-B0292A
CAS No.: 64228-81-5
Synonyms: BW-33A
Target:  

nAChR

Atracurium (BW-33A) besylate is a potent, competitive and non-depolarizing neuromuscular blocking agent. Atracurium besylate also is an AChR receptor antagonist. Atracurium besylate induces bronchoconstriction and neuromuscular blockade. Atracurium besylate promotes astroglial differentiation .
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Cat. No.: HY-122140
CAS No.: 795316-16-4
Purity:  99.72%
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

ACG548B (compound 24) is a potent inhibitor of acetyl- and butyrylcholinesterase (AChE and BChE) with IC50s of 1.78 and 0.496 μM, respectively. ACG548B has higher AChE affinity and selectivity over BChE and ChoK (choline kinase). ACG548B can be uesd for the study of myasthenia gravis and neuromuscular blockade .
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Cat. No.: HY-159818
CAS No.: 1309580-40-2
Synonyms: Adamgammadex; Aom0498
Target:  

Drug Derivative

Research Areas:  

Neurological Disease

Amogammadex (Adamgammadex; Aom0498) is a modified γ-cyclodextrin (HY-W040040) derivative and neuromuscular blocking agent. Amogammadex forms inactive, tight inclusion complexes with free Rocuronium (HY-17033) and Vecuronium (HY-B0118A), and reverses the neuromuscular blockade induced by them in a concentration-dependent manner. Amogammadex can be used in research related to neuromuscular blockade reversal .
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Cat. No.: HY-B0292
CAS No.: 64228-79-1
Synonyms: BW-33A free acid
tracurium (BW-33A free acid) is a potent, competitive and non-depolarizing neuromuscular blocking agent.Atracurium also is an AChR receptor antagonist. Atracurium induces bronchoconstriction and neuromuscular blockade. Atracurium promotes astroglial differentiation .
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Cat. No.: HY-B0292AR
CAS No.: 64228-81-5
Synonyms: BW-33A (Standard)
Atracurium (besylate) (Standard) is the analytical standard of Atracurium (besylate). This product is intended for research and analytical applications. Atracurium (BW-33A) besylate is a potent, competitive and non-depolarizing neuromuscular blocking agent. Atracurium besylate also is an AChR receptor antagonist. Atracurium besylate induces bronchoconstriction and neuromuscular blockade. Atracurium besylate promotes astroglial differentiation .
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Cat. No.: HY-124047
CAS No.: 40709-76-0
Target:  

Cholinesterase (ChE)

Research Areas:  

Neurological Disease

RX 67668 is a potent cholinesterase inhibitor with an IC50 of 5 μM for both acetylcholinesterase (AChE) and butyrylcholinesterase. RX 67668 can reverse the neuromuscular blockade induced by D-tubocurarine. RX 67668 is a muscle relaxant used to relieve skeletal muscle fatigue .
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Cat. No.: HY-182537
CAS No.: 119302-18-0
Target:  

Drug Derivative

Research Areas:  

Neurological Disease

Org 9616 bromide is a non-depolarizing neuromuscular blocker with a structure similar to Pancuroniam. Org 9616 bromide induces rapid-onset, short-duration neuromuscular blockade .
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Cat. No.: HY-127147
CAS No.: 49564-56-9
Synonyms: AH 8165 bromide
Target:  

mAChR

Research Areas:  

Neurological Disease

Fazadinium bromide (AH 8165 bromide) is a species-specific neuromuscular blocking agent that primarily targets the acetylcholine receptor (AChR) at the skeletal neuromuscular junction, blocking the receptor agonist binding site in a competitive and reversible manner. Fazadinium bromide induces sustained tetanic fade, and tetanic contractions are more sensitive than single twitches. Fazadinium bromide can be used in anesthesia and research related to neuromuscular transmission .
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