Idalopirdine Hydrochloride (Synonyms: Lu AE58054 (Hydrochloride))

Cat. No.: HY-14338A Purity: 99.17%
Handling Instructions

Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is a potent and selective 5-HT6 receptor antagonist with a Ki of 0.83 nM.

For research use only. We do not sell to patients.

Idalopirdine Hydrochloride Chemical Structure

Idalopirdine Hydrochloride Chemical Structure

CAS No. : 467458-02-2

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 290 In-stock
Estimated Time of Arrival: December 31
5 mg USD 264 In-stock
Estimated Time of Arrival: December 31
10 mg USD 403 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1087 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
200 mg   Get quote  

* Please select Quantity before adding items.

Other Forms of Idalopirdine Hydrochloride:

  • Biological Activity

  • Technical Information

  • Purity & Documentation

Description

Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is a potent and selective 5-HT6 receptor antagonist with a Ki of 0.83 nM.

Clinical Trial
Solvent & Solubility
In Vitro: 

DMSO : ≥ 25 mg/mL (57.49 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.2997 mL 11.4987 mL 22.9975 mL
5 mM 0.4599 mL 2.2997 mL 4.5995 mL
10 mM 0.2300 mL 1.1499 mL 2.2997 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.5 mg/mL (5.75 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.5 mg/mL (5.75 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.5 mg/mL (5.75 mM); Clear solution

Molecular Weight

434.83

Formula

C₂₀H₂₀ClF₅N₂O

CAS No.

467458-02-2

SMILES

FC1=CC(NC=C2CCNCC3=CC(OCC(F)(F)C(F)F)=CC=C3)=C2C=C1.Cl

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
Idalopirdine Hydrochloride
Cat. No.:
HY-14338A
Quantity:

Idalopirdine Hydrochloride

Cat. No.: HY-14338A