1. Signaling Pathways
  2. GPCR/G Protein
  3. Amylin Receptor
  4. Amylin Receptor Antagonist

Amylin Receptor Antagonist

Amylin Receptor Antagonists (7):

Cat. No. Product Name Effect Purity
  • HY-P10745
    Petrelintide
    Antagonist 99.49%
    Petrelintide (ZP8396) is a dual amylin and calcitonin receptor agonist (DACRA) Petrelintide elicits a selective reduction in high-fat diet intake in diet-induced obese (DIO) rats, which is accompanied by a loss of fat mass and preservation of lean mass during weight reduction. Petrelintide can be utilized in diabetes research.
  • HY-P10745A
    Petrelintide acetate
    Antagonist 99.81%
    Perelintide (ZP8396) acetate is a dual amylin and calcitonin receptor agonist (DACRA). Perelintide acetate elicits a selective reduction in high-fat diet intake in diet-induced obese (DIO) rats, which is accompanied by a loss of fat mass and preservation of lean mass during weight reduction. Perelintide acetate can be utilized in diabetes research.
  • HY-P1782
    Calcitonin (8-32), salmon
    Antagonist 99.81%
    Calcitonin (8-32), salmon is a highly selective Amylin receptor antagonist. Calcitonin (8-32), salmon reverses the Amylin-mediated inhibition of glucose-induced insulin release, but has no effect on either glucagon release or somatostatin release. Calcitonin (8-32), salmon can be used for studies related to β-cell amylin.
  • HY-P10235
    Cyclic AC253
    Antagonist 99.83%
    Cyclic AC253 is an antagonist for amylin receptor, with IC50 of 0.3 μM. Cyclic AC253 exhibits neuroprotective efficacy against Aβ toxicity and abrogates Aβ-induced impairment of hippocampal long-term potentiation. Cyclic AC253 penetrate blood-brain barrier (BBB).
  • HY-P4928
    Biotinyl-Amylin (mouse, rat)
    Antagonist 99.89%
    Biotinyl-Amylin (mouse, rat) is a biotinylated Amylin (mouse, rat). Amylin (mouse, rat) is a 37-aminoacid pancreatic protein that exerts control over several metabolic events such as glycemia and lacticemia.
  • HY-P4785
    Acetyl-Amylin (8-37) (human)
    Antagonist
    Acetyl-Amylin (8-37) (human) is a specific amylin antagonist.
  • HY-P4928A
    Biotinyl-Amylin (mouse, rat) TFA
    Antagonist
    Biotinyl-Amylin (mouse, rat) TFA is a biotinylated Amylin (mouse, rat). Amylin (mouse, rat) is a 37-aminoacid pancreatic protein that exerts control over several metabolic events such as glycemia and lacticemia.