1253919-92-4
Chemical Structure
CH5447240
- CAS No.: 1253919-92-4
- Formula:C26H39N5O4S
- Molecular Weight:517.68
IUPAC Name: 1-(3,5-dimethyl-4-(2-((2-((1r,4r)-4-methylcyclohexyl)-4-oxo-1,3,8-triazaspiro[4.5]dec-2-en-8-yl)sulfonyl)ethyl)phenyl)-1-methylurea
InChIKey: PNTBFOBXKXSPLI-IRJFHVNHSA-N
SMILES: O=C(N)N(C1=CC(C)=C(CCS(=O)(N(CC2)CCC2(NC([C@H]3CC[C@H](C)CC3)=N4)C4=O)=O)C(C)=C1)C
Biological Activity: CH5447240 is an agonist for parathyroid hormone receptor 1 (PTHR1), that inhibits human PTHR1 with an EC50 of 12 μM. CH5447240 exhibits good metabolic stability in human liver microsomes. CH5447240 increases serum calcium levels in rats. CH5447240 can be used in research about hypoparathyroidism[1].
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CH5447240 | CH5447240 is an agonist for parathyroid hormone receptor 1 (PTHR1), that inhibits human PTHR1 with an EC50 of 12 μM. CH5447240 exhibits good metabolic stability in human liver microsomes. CH5447240 increases serum calcium levels in rats. CH5447240 can be used in research about hypoparathyroidism. | |||||||||||||||||||||
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Keywords
