134208-17-6
Chemical Structure
Mazapertine
- CAS No.: 134208-17-6
- Formula:C26H35N3O2
- Molecular Weight:421.58
IUPAC Name: (3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)phenyl)(piperidin-1-yl)methanone
InChIKey: ZKZFPRUSWCYSGT-UHFFFAOYSA-N
SMILES: CC(C)OC1=C(N2CCN(CC3=CC(C(N4CCCCC4)=O)=CC=C3)CC2)C=CC=C1
Biological Activity: Mazapertine is an orally active antipsychotic agent. M azapertine antagonizes to dopamine D2/3/4 receptors (Ki values < 3 nM) and also strongly binds to serotonin 5-HT1A receptor (Ki =1.7 nM) and α1-adrenergic receptor (Ki = 1.3 nM). Mazapertine can be used for the research of neurological disease[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Mazapertine | 99.37% | Mazapertine is an orally active antipsychotic agent. M azapertine antagonizes to dopamine D2/3/4 receptors (Ki values < 3 nM) and also strongly binds to serotonin 5-HT1A receptor (Ki =1.7 nM) and α1-adrenergic receptor (Ki = 1.3 nM). Mazapertine can be used for the research of neurological disease. | ||||||||||||||||||||
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Keywords
