1422053-03-9
1422053-03-9
Chemical Structure
TMP780
- CAS No.: 1422053-03-9
- Formula:C31H30N2O4
- Molecular Weight:494.58
IUPAC Name: 2-(2-((R)-(3,5-dimethylisoxazol-4-yl)(hydroxy)methyl)benzofuran-5-yl)-N-((S)-(2,4-dimethylphenyl)(phenyl)methyl)acetamide
InChIKey: DIURRJOJDQOMFC-CONSDPRKSA-N
SMILES: O=C(N[C@H](C1=CC=C(C)C=C1C)C2=CC=CC=C2)CC3=CC=C(OC([C@@H](C4=C(C)ON=C4C)O)=C5)C5=C3
Biological Activity: TMP780 is an inverse agonist of RORγt with an IC50 of 13 nM. RORγt is a tractable agent target for the treatment of cutaneous inflammatory disorders[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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TMP780 | 99.51% | TMP780 is an inverse agonist of RORγt with an IC50 of 13 nM. RORγt is a tractable agent target for the treatment of cutaneous inflammatory disorders. | ||||||||||||||||||||
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TMP780 (Standard) | ≥98% | TMP780 (Standard) is the analytical standard of TMP780 (HY-102075B). This product is intended for research and analytical applications. TMP780 is an inverse agonist of RORγt with an IC50 of 13 nM. RORγt is a tractable agent target for the treatment of cutaneous inflammatory disorders. | ||||||||||||||||||||
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References
Keywords
