1841464-21-8
1841464-21-8
Chemical Structure
K-Ras-PDEδ-IN-1
- CAS No.: 1841464-21-8
- Formula:C25H26FN5O2
- Molecular Weight:447.50
IUPAC Name: N-(4-fluorophenethyl)-4-(4-methyl-7-oxo-2-(p-tolyl)-2,7-dihydro-6H-pyrazolo[3,4-d]pyridazin-6-yl)butanamide
InChIKey: RRELLHHWESTKAK-UHFFFAOYSA-N
SMILES: O=C(NCCC1=CC=C(F)C=C1)CCCN2N=C(C)C3=CN(C4=CC=C(C)C=C4)N=C3C2=O
Biological Activity: K-Ras-PDEδ-IN-1 is a novel and potent competitive K-Ras-PDEδ inhibitor. K-Ras-PDEδ-IN-1 binds to the farnesyl binding pocket of PDEδ with a low nanomolar Kd of 8 nM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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K-Ras-PDEδ-IN-1 | 99.45% | K-Ras-PDEδ-IN-1 is a novel and potent competitive K-Ras-PDEδ inhibitor. K-Ras-PDEδ-IN-1 binds to the farnesyl binding pocket of PDEδ with a low nanomolar Kd of 8 nM. | ||||||||||||||||||||
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References
Keywords
