2250024-74-7
2250024-74-7
Chemical Structure
DDO-2093
- CAS No.: 2250024-74-7
- Formula:C29H37ClFN9O3
- Molecular Weight:614.11
IUPAC Name: 1-(3-(5-amino-2-chloro-4-fluoro-3-methylbenzamido)-4-(4-methylpiperazin-1-yl)phenyl)-N-(3-morpholinopropyl)-1H-1,2,3-triazole-4-carboxamide
InChIKey: MPTAUAHHFUFKAG-UHFFFAOYSA-N
SMILES: O=C(C1=CN(C2=CC=C(N3CCN(C)CC3)C(NC(C4=CC(N)=C(F)C(C)=C4Cl)=O)=C2)N=N1)NCCCN5CCOCC5
Biological Activity: DDO-2093 is a potent MLL1-WDR5 protein-protein interaction inhibitor (IC50=8.6 nM; Kd=11.6 nM) with antitumor activity. DDO-2093 selectively inhibits the catalytic activity of MLL complex[1].
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DDO-2093 | DDO-2093 is a potent MLL1-WDR5 protein-protein interaction inhibitor (IC50=8.6 nM; Kd=11.6 nM) with antitumor activity. DDO-2093 selectively inhibits the catalytic activity of MLL complex. | |||||||||||||||||||||
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References
Keywords
