2374971-81-8
2374971-81-8
Chemical Structure
CPI-1612
- CAS No.: 2374971-81-8
- Formula:C27H26N6O
- Molecular Weight:450.53
IUPAC Name: (R)-2-(((S)-2-(4-cyanophenyl)propyl)amino)-N-(5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl)-2-phenylacetamide
InChIKey: SEDFZSHSBUXKAC-NIYFSFCBSA-N
SMILES: O=C(NC1=NC=C(C2=CN(C)N=C2)C=C1)[C@H](NC[C@H](C3=CC=C(C#N)C=C3)C)C4=CC=CC=C4
Biological Activity: CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CPI-1612 | 99.75% | CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity. | ||||||||||||||||||||
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References
Keywords
