2413257-74-4
2413257-74-4
Chemical Structure
A3AR antagonist 1
- CAS No.: 2413257-74-4
- Formula:C32H24N4O4S
- Molecular Weight:560.62
IUPAC Name: 4-methoxy-N-(5-(3-(4-methoxyphenyl)-4-oxo-3,4-dihydroquinazolin-2-yl)-4-phenylthiazol-2-yl)benzamide
InChIKey: UFKAMNUQGBWBJM-UHFFFAOYSA-N
SMILES: COC1=CC=C(C=C1)C(NC2=NC(C3=CC=CC=C3)=C(S2)C4=NC5=C(C(N4C6=CC=C(C=C6)OC)=O)C=CC=C5)=O
Biological Activity: A3AR antagonist 1 (compound 17) is a potent and selective human A3 adenosine receptor (AR) antagonist, with an Ki of 4.63 nM. A3AR antagonist 1 shows no affinity for the rat A3 AR even at high concentrations[1].
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A3AR antagonist 1 | A3AR antagonist 1 (compound 17) is a potent and selective human A3 adenosine receptor (AR) antagonist, with an Ki of 4.63 nM. A3AR antagonist 1 shows no affinity for the rat A3 AR even at high concentrations. | |||||||||||||||||||||
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References
Keywords
