A3AR antagonist 1
A3AR antagonist 1 (compound 17) is a potent and selective human A3 adenosine receptor (AR) antagonist, with an Ki of 4.63 nM. A3AR antagonist 1 shows no affinity for the rat A3 AR even at high concentrations.
For research use only. We do not sell to patients.
- CAS No.: 2413257-74-4
- Formula: C32H24N4O4S
- Molecular Weight:560.62
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adenosine Receptor Isoforms
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Biological Activity
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hA3 4.63 nM (Ki) |
Chemical Information
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CAS No. 2413257-74-4
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Molecular Weight 560.62
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Formula C32H24N4O4S
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SMILES
COC1=CC=C(C=C1)C(NC2=NC(C3=CC=CC=C3)=C(S2)C4=NC5=C(C(N4C6=CC=C(C=C6)OC)=O)C=CC=C5)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)