2641595-55-1
2641595-55-1
Chemical Structure
Bivamelagon hydrochloride
Synonym(s): MC-4R Agonist 2 hydrochloride
- CAS No.: 2641595-55-1
- Formula:C35H54Cl2N4O4
- Molecular Weight:665.73
InChIKey: DPMKLJUIFGHPGV-MVCZUIQNSA-N
SMILES: O=C([C@H]1[C@H](C2=CC=C(C=C2)Cl)CN(C1)C(C)(C)C)N3[C@@H](C[C@@H](C3)N([C@@H]4CC[C@@H](CC4)C)C(C(C)C)=O)C(N5CCOCC5)=O.[H]Cl
Biological Activity: Bivamelagon (MC-4R Agonist 2) hydrochloride is an orally active and BBB-penetrable MC4R agonist with EC50 values of 0.562 nM (Luci assay) and 36.5 nM (cAMP assay), and a Ki of 65 nM. Bivamelagon hydrochloride can be used for the research of diseases such as obesity and diabetes[1].
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Bivamelagon hydrochloride | Bivamelagon (MC-4R Agonist 2) hydrochloride is an orally active and BBB-penetrable MC4R agonist with EC50 values of 0.562 nM (Luci assay) and 36.5 nM (cAMP assay), and a Ki of 65 nM. Bivamelagon hydrochloride can be used for the research of diseases such as obesity and diabetes. | |||||||||||||||||||||
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