2761281-51-8
2761281-51-8
Chemical Structure
PROTAC(H-PGDS)-8
- CAS No.: 2761281-51-8
- Formula:C41H40N8O7
- Molecular Weight:756.81
InChIKey: UUILKUWMNHXPIN-UHFFFAOYSA-N
SMILES: O=C(C1CCN(CC1)C2=CC=C(C=C2)NC(C3=CN=C(N=C3)OC4=CC=CC=C4)=O)N5CCN(CC5)C6=C(C7=CC=C6)C(N(C7=O)C8CCC(N(C8=O)C)=O)=O
Biological Activity: PROTAC (H-PGDS)-8 is an H-PGDS PROTAC inhibitor with a IC50 of 0.14 μM. PROTAC (H-PGDS)-8 binds to H-PGDS and inhibits its enzymatic activity. PROTAC (H-PGDS)-8 inhibits the production of PGD2 in cancer cells. PROTAC (H-PGDS)-8 can be used for the research of Duchenne muscular dystrophy[1].
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PROTAC(H-PGDS)-8 | PROTAC (H-PGDS)-8 is an H-PGDS PROTAC inhibitor with a IC50 of 0.14 μM. PROTAC (H-PGDS)-8 binds to H-PGDS and inhibits its enzymatic activity. PROTAC (H-PGDS)-8 inhibits the production of PGD2 in cancer cells. PROTAC (H-PGDS)-8 can be used for the research of Duchenne muscular dystrophy. | |||||||||||||||||||||
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References
Keywords
