2767560-94-9
2767560-94-9
Chemical Structure
A2AAR/HDAC-IN-2
- CAS No.: 2767560-94-9
- Formula:C23H26N6O4
- Molecular Weight:450.49
IUPAC Name: 7-(3-((6-amino-4-(furan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)phenoxy)-N-hydroxyheptanamide
InChIKey: BNMVLBFIXXFEJN-UHFFFAOYSA-N
SMILES: NC1=NC(C2=CC=CO2)=C3C=NN(C3=N1)CC4=CC=CC(OCCCCCCC(NO)=O)=C4
Biological Activity: A2AAR/HDAC-IN-2 is a potent A2AAR/HDAC dual inhibitor, with good binding affinity for A2AAR (Ki=10.3 nM) and good inhibitory activity against HDAC1 (IC50=18.5 nM). A2AAR/HDAC-IN-2 can be used in study of antitumor[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
A2AAR/HDAC-IN-2 | A2AAR/HDAC-IN-2 is a potent A2AAR/HDAC dual inhibitor, with good binding affinity for A2AAR (Ki=10.3 nM) and good inhibitory activity against HDAC1 (IC50=18.5 nM). A2AAR/HDAC-IN-2 can be used in study of antitumor. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
