288150-92-5
288150-92-5
Chemical Structure
SB-408124
- CAS No.: 288150-92-5
- Formula:C19H18F2N4O
- Molecular Weight:356.37
IUPAC Name: 1-(6,8-difluoro-2-methylquinolin-4-yl)-3-(4-(dimethylamino)phenyl)urea
InChIKey: JTARFZSNUAGHRB-UHFFFAOYSA-N
SMILES: O=C(NC1=CC(C)=NC2=C(C=C(C=C21)F)F)NC3=CC=C(C=C3)N(C)C
Biological Activity: SB-408124 is a non-peptide OX1 receptor antagonist with Kis of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 exhibits 50-fold selectivity over OX2 receptor[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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SB-408124 | 98.93% | SB-408124 is a non-peptide OX1 receptor antagonist with Kis of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 exhibits 50-fold selectivity over OX2 receptor. | ||||||||||||||||||||
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SB-408124 (Standard) | ≥98% | SB-408124 (Standard) is the analytical standard of SB-408124. This product is intended for research and analytical applications. SB-408124 is a non-peptide OX1 receptor antagonist with Kis of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 exhibits 50-fold selectivity over OX2 receptor. | ||||||||||||||||||||
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References
Keywords
