2941268-96-6
2941268-96-6
Chemical Structure
ERα degrader 5
- CAS No.: 2941268-96-6
- Formula:C29H25F4N3O2S
- Molecular Weight:555.59
IUPAC Name: 2-(2-(1,1-difluoroethyl)-4-fluorophenyl)-3-(4-((1-(3-fluoropropyl)azetidin-3-yl)oxy)phenoxy)-6H-thieno[2,3-e]indazole
InChIKey: QGTNFUUVOBBVAM-UHFFFAOYSA-N
SMILES: CC(F)(C1=C(C2=C(C3=CC=C4NN=CC4=C3S2)OC5=CC=C(C=C5)OC6CN(C6)CCCF)C=CC(F)=C1)F
Biological Activity: ERα degrader 5 (Compound 40) is a selective, orally bioavailable estrogen receptor (ER) degrader (SERD) with an EC50 of 1.1 nM against ERα. ERα degrader 5 shows antitumor effect in vivo[1].
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ERα degrader 5 | ERα degrader 5 (Compound 40) is a selective, orally bioavailable estrogen receptor (ER) degrader (SERD) with an EC50 of 1.1 nM against ERα. ERα degrader 5 shows antitumor effect in vivo. | |||||||||||||||||||||
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References
Keywords
