2971825-58-6
2971825-58-6
Chemical Structure
α2A-AR agonist 1
- CAS No.: 2971825-58-6
- Formula:C12H11BrN2O
- Molecular Weight:279.13
InChIKey: CDYNCVBGLQHJIS-UHFFFAOYSA-N
SMILES: BrC1=C(C2=CC=C1)OCCC2C3=CNC=N3
Biological Activity: α2A-AR agonist 1 (Compound B9) is a selective agonist for α2-adrenergic receptor (α2A-AR) with EC50 of 0.23 nM. α2A-AR agonist 1 exhibits a hypnotic effect, with ED50 of 0.138 mg/kg in the loss of righting reflex (LORR) experiment. α2A-AR agonist 1 exhibits metabolic stability in mouse liver microsomes[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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α2A-AR agonist 1 | 99.92% | α2A-AR agonist 1 (Compound B9) is a selective agonist for α2-adrenergic receptor (α2A-AR) with EC50 of 0.23 nM. α2A-AR agonist 1 exhibits a hypnotic effect, with ED50 of 0.138 mg/kg in the loss of righting reflex (LORR) experiment. α2A-AR agonist 1 exhibits metabolic stability in mouse liver microsomes. | ||||||||||||||||||||
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References
Keywords
