302826-61-5

EPAC 5376753 Chemical Structure
302826-61-5

Chemical Structure

EPAC 5376753

  • CAS No.: 302826-61-5
  • Formula:C15H8Cl2N2O3S
  • Molecular Weight:367.21

IUPAC Name: 5-((5-(2,4-dichlorophenyl)furan-2-yl)methylene)-2-thioxodihydropyrimidine-4,6(1H,5H)-dione

InChIKey: QQAOFKJHOUFHKI-UHFFFAOYSA-N

SMILES: O=C(/C(C(N1)=O)=C/C2=CC=C(C3=CC=C(Cl)C=C3Cl)O2)NC1=S

Biological Activity: EPAC 5376753, a 2-Thiobarbituric acid (HY-77962) derivative, is a selective and allosteric Epac inhibitor. EPAC 5376753 inhibits Epac1 with an IC50 of 4 µM in Swiss 3T3 cells. EPAC 5376753 does not inhibit PKA and adenylyl cyclases[1].

Cat. No. Product Name Purity Description Pricing
HY-111446 		EPAC 5376753 98.10% EPAC 5376753, a 2-Thiobarbituric acid (HY-77962) derivative, is a selective and allosteric Epac inhibitor. EPAC 5376753 inhibits Epac1 with an IC50 of 4 µM in Swiss 3T3 cells. EPAC 5376753 does not inhibit PKA and adenylyl cyclases.
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