3050872-68-6
3050872-68-6
Chemical Structure
CBP/BRD4-IN-1
- CAS No.: 3050872-68-6
- Formula:C39H53N5O5
- Molecular Weight:671.87
InChIKey: YGDLXRXBIULMJO-UHFFFAOYSA-N
SMILES: CCN(C1=CC(C2=CC=C(CN3CCN(CCC(O)=O)CC3)C=C2)=CC(C(N(CC4=C(C=C(N(C4=O)C)C)C)C)=O)=C1C)C5CCOCC5
Biological Activity: CBP/BRD4-IN-1 (Compound 22) is a dual bromodomain inhibitor of CBP and BRD4 BD1, with IC50 values of 1.2 μM and 3.2 μM, respectively. CBP/BRD4-IN-1 serves as a target protein ligand for the synthesis of PROTACs, such as MS8847N1 (HY-18626)[1].
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CBP/BRD4-IN-1 | CBP/BRD4-IN-1 (Compound 22) is a dual bromodomain inhibitor of CBP and BRD4 BD1, with IC50 values of 1.2 μM and 3.2 μM, respectively. CBP/BRD4-IN-1 serves as a target protein ligand for the synthesis of PROTACs, such as MS8847N1 (HY-18626). | |||||||||||||||||||||
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References
Keywords
