CBP/BRD4-IN-1
CBP/BRD4-IN-1 (Compound 22) is a dual bromodomain inhibitor of CBP and BRD4 BD1, with IC50 values of 1.2 μM and 3.2 μM, respectively. CBP/BRD4-IN-1 serves as a target protein ligand for the synthesis of PROTACs, such as MS8847N1 (HY-18626).
For research use only. We do not sell to patients.
- CAS No.: 3050872-68-6
- Formula: C39H53N5O5
- Molecular Weight:671.87
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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CBP 1.2 μM (IC50) |
BRD4 3.2 μM (IC50) |
EZH2 |
Chemical Information
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CAS No. 3050872-68-6
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Molecular Weight 671.87
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Formula C39H53N5O5
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SMILES
CCN(C1=CC(C2=CC=C(CN3CCN(CCC(O)=O)CC3)C=C2)=CC(C(N(CC4=C(C=C(N(C4=O)C)C)C)C)=O)=C1C)C5CCOCC5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CBP/BRD4-IN-1 Related Classifications
HY-186270 Related Classifications
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