CBP/BRD4-IN-1
CBP/BRD4-IN-1 (Compound 22) is a dual bromodomain inhibitor of CBP and BRD4 BD1, with IC50 values of 1.2 μM and 3.2 μM, respectively. CBP/BRD4-IN-1 serves as a target protein ligand for the synthesis of PROTACs, such as MS8847N1 (HY-18626).
Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.
- CAS No.: 3050872-68-6
- Formule: C39H53N5O5
- Masse moléculaire:671.87
-
Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Activité biologique
-
Chemical Information
- Pureté et documentation
- Références
-
Help & FAQs
Activité biologique
Description
IC50 & Target
[1]|
CBP 1.2 μM (IC50) |
BRD4 3.2 μM (IC50) |
EZH2 |
Chemical Information
-
CAS No. 3050872-68-6
-
Masse moléculaire 671.87
-
Formule C39H53N5O5
-
SMILES
CCN(C1=CC(C2=CC=C(CN3CCN(CCC(O)=O)CC3)C=C2)=CC(C(N(CC4=C(C=C(N(C4=O)C)C)C)C)=O)=C1C)C5CCOCC5
-
Livraison
Room temperature in continental US; may vary elsewhere.
-
Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CBP/BRD4-IN-1 Related Classifications
HY-186270 Related Classifications
Powered by Bioz