3086024-48-5
3086024-48-5
Chemical Structure
CBP/p300/BRD4 ligand-1
- CAS No.: 3086024-48-5
- Formula:C22H25F3N4O2
- Molecular Weight:434.45
InChIKey: CJZXLBCBVDPIOI-UHFFFAOYSA-N
SMILES: CC1=CC(C(C=C2N3CCOC(F)(F)F)=CC=C2N=C3C4CCNCC4)=CN(C1=O)C
Biological Activity: CBP/p300/BRD4 ligand-1 is a small-molecule inhibitor targeting CBP, p300, and BRD4. CBP/p300/BRD4 ligand-1 competitively binds to the functional domains of target proteins without disrupting key interactions. CBP/p300/BRD4 ligand-1 can be used for the construction of dual-target PROTAC degraders (HY-181758) in studies related to prostate cancer and other cancers[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
CBP/p300/BRD4 ligand-1 | CBP/p300/BRD4 ligand-1 is a small-molecule inhibitor targeting CBP, p300, and BRD4. CBP/p300/BRD4 ligand-1 competitively binds to the functional domains of target proteins without disrupting key interactions. CBP/p300/BRD4 ligand-1 can be used for the construction of dual-target PROTAC degraders (HY-181758) in studies related to prostate cancer and other cancers. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
