380620-88-2
![[(pF)Phe4]Nociceptin(1-13)NH2 Chemical Structure](http://file.medchemexpress.cn/product_pic/hy-p1300.gif "[(pF)Phe4]Nociceptin(1-13)NH2 Chemical Structure")
380620-88-2
Chemical Structure
[(pF)Phe4]Nociceptin(1-13)NH2
- CAS No.: 380620-88-2
- Formula:C61H99FN22O15
- Molecular Weight:1399.58
SMILES: [FGG{Phe(4-F)}TGARKSARK-NH2]
Biological Activity: [(pF)Phe4]Nociceptin(1-13)NH2 is a highly potent and selective NOP receptor (OP4) agonist, with a pKi of 10.68 and a pEC50 of 9.31. [(pF)Phe4]Nociceptin(1-13)NH2 displays high selectivity over δ, κ, and μ opioid receptors (>3000 fold)[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
[(pF)Phe4]Nociceptin(1-13)NH2 | [(pF)Phe4]Nociceptin(1-13)NH2 is a highly potent and selective NOP receptor (OP4) agonist, with a pKi of 10.68 and a pEC50 of 9.31. [(pF)Phe4]Nociceptin(1-13)NH2 displays high selectivity over δ, κ, and μ opioid receptors (>3000 fold). | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
- [1]. Rizzi A, et al. Pharmacological characterisation of [(pX)Phe4]nociceptin(1-13)NH2 analogues. 2. In vivo studies. Naunyn Schmiedebergs Arch Pharmacol. 2002;365(6):450-456. [Content Brief]
- [2]. Bigoni R, et al. Pharmacological characterisation of [(pX)Phe4]nociceptin(1-13)amide analogues. 1. In vitro studies. Naunyn Schmiedebergs Arch Pharmacol. 2002;365(6):442-449. [Content Brief]
Keywords
