HCN2 modulator-4
HCN2 modulator-4 is a HCN2 ion channel inhibitor. HCN2 modulator-4 inhibits HCN2 ion channel activity. HCN2 modulator-4 can be used for the research of pain, inflammatory pain, neuropathic pain, tinnitus, central nervous system disorders, psychiatric disorders, mood disorders.
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- CAS No.: 3080809-03-3
- Formule: C23H21FN4O5
- Masse moléculaire:452.44
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
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KCNQ2 |
HCN2 modulator-4 (R-configuration 39; 5 minutes) potently inhibits human HCN2 channels with an IC50 of 10 nM, with reduced activity against human HCN1 and HCN4 channels[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3080809-03-3
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Masse moléculaire 452.44
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Formule C23H21FN4O5
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SMILES
O=C(C1=C(OC=C1)C)NC2=NN(C[C@@H](C)OC)C3=NC=C(C4=CC(F)=C(OCO5)C5=C4)C=C23
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)