Pecavaptan
Pecavaptan, a chemical probe, is an orally active and dual antagonist of V1a/V2 receptor (Ki=0.5 nM and 0.6 nM for human, respectively). Pecavaptan promotes an increase in urine production, which reduces the associated symptoms of water retention and edema.
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- No. CAS: 1914998-56-3
- Fòrmula: C22H19Cl2F3N6O3
- Peso molecular:543.33
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Actividad biológica
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Chemical Information
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Help & FAQs
Ver todos los productos específicos de isoformas Vasopressin Receptor
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Actividad biológica
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human V1a Receptor 3.6 nM (IC50) |
canine V1a Receptor 4.4 nM (IC50) |
human V2 Receptor 1.7 nM (IC50) |
canine V2 Receptor 1.3 nM (IC50) |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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No. CAS 1914998-56-3
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Peso molecular 543.33
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Fòrmula C22H19Cl2F3N6O3
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SMILES
O[C@H](C(F)(F)F)CN1C(C2=CC=C(Cl)C=C2)=NN(CC3=NN(C4=CC(Cl)=CC=C4)C([C@@H](O)C)=N3)C1=O
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Synonyms
BAY 1753011
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Pecavaptan Related Classifications
HY-109133 Related Classifications
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