1 Result for "

(Rac)-AMG8379

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "(Rac)-AMG8379" in MCE Product Catalog:

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Cat. No.: HY-108425B
CAS No.: 1641574-26-6
Synonyms: (Rac)-AMG8380
Target:  

Sodium Channel

Research Areas:  

Neurological Disease

(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379. AMG8379 is a potent, orally active and selective sulfonamide antagonist of NaV1.7, with IC50s of 8.5 and 18.6 nM for hNaV1.7 and mNaV1.7, respectively .
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