1 Result for "

2376991-14-7

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "2376991-14-7" in MCE Product Catalog:

Cat. No.: HY-176955
CAS No.: 2376991-14-7
Target:  

Estrogen Receptor/ERR

Research Areas:  

Cancer

ER degrader 12 (Example 1) is an estrogen receptor (ER) degrader with IC50 values for ERα and ERβ of 2.3 and 80.2 nM respectively (TR-FRET experiment). ER degrader 12 inhibits the proliferation of MCF-7 cells, with an IC50 of 1.53 nM. ER degrader 12 can be used for research on breast cancer .
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