1 Result for "

2566733-45-5

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "2566733-45-5" in MCE Product Catalog:

Cat. No.: HY-168439
CAS No.: 2566733-45-5
HLB-0532259 is a Aurora-A/N-Myc PROTAC degrader, with a DC50 of 20.2 nM against Aurora-A in MCF-7 cells; its DC50 values against N-Myc are 179 nM in SK-N-BE (2) cells and 229 nM in Kelly cells, respectively. HLB-0532259 induces apoptosis (apoptosis) in MYCN-amplified neuroblastoma cells and inhibits tumor growth in mouse xenograft models. HLB-0532259 can be used for the research of neuroblastoma .
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