1 Result for "

2586195-28-8

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "2586195-28-8" in MCE Product Catalog:

Cat. No.: HY-146494
CAS No.: 2586195-28-8
Target:  

Androgen Receptor

Research Areas:  

Cancer

Androgen receptor antagonist 5 (compound 42f) is a potent androgen receptor (AR) antagonist with an IC50 value of 6.17 μM. Androgen receptor antagonist 5 can effectively impair AR nuclear translocation, reducing the levels of nuclear AR, and disrupts AR-mediated gene regulation. Androgen receptor antagonist 5 has antiproliferative activity against LNCaP and exhibits antitumor activity in LNCaP xenograft tumor mice model. Androgen receptor antagonist 5 can be used for researching prostate cancer .
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