1 Result for "

3030279-55-8

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "3030279-55-8" in MCE Product Catalog:

Cat. No.: HY-175842
CAS No.: 3030279-55-8
Target:  

PROTACs CDK

Research Areas:  

Cancer

PROTAC CDK2 Degrader-2 is an orally active CDK2 PROTAC degrader, with DC50 values of 13 nM (MKN1cells) and 17 nM (TOV21G cells). PROTAC CDK2 Degrader-2 induces G1 phase arrest in MKN1 cells. PROTAC CDK2 Degrader-2 achieves tumor stasis in HCC1569 (CCNE1-amplified) xenograft models. PROTAC CDK2 Degrader-2 can be used for the study of CCNE1-amplified cancers .
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