1 Result for "

3036457-38-9

" in MedChemExpress (MCE) Product Catalog:
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1 Results for "3036457-38-9" in MCE Product Catalog:

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1 Cited Publications
Cat. No.: HY-155994
CAS No.: 3036457-38-9
Purity:  99.90%
Target:  

PROTACs PIKfyve Autophagy

Research Areas:  

Cancer

PIK5-12d is a PROTAC PIKfyve degrader (DC50 = 1.48 nM). PIK5-12d induces massive cytoplasmic vacuolization and blocks autophagic flux in multiple prostate cancer cells. PIK5-12d inhibits prostate cancer cell proliferation. PIK5-12d significantly suppresses tumor proliferation in mice bearing LTL-331R human prostate cancer PDX tumors. PIK5-12d can be used for the study of prostate cancer .
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